Compound Profile: Dezlorid
Dezlorid 5 mg is a pharmaceutical-grade desloratadine preparation manufactured by Intas Pharmaceuticals for in-vitro laboratory research. Desloratadine is a third-generation tricyclic antihistamine compound classified as a selective histamine H1 receptor antagonist. This non-sedating antihistamine demonstrates high binding affinity for peripheral H1 receptors while exhibiting minimal central nervous system penetration in preclinical models. Researchers at Stroid UK Shop investigate desloratadine’s pharmacological properties in histamine-mediated inflammatory response studies and allergic pathway research.
Laboratory Applications
Research teams examine desloratadine’s mechanism of action as a selective antagonist of histamine H1 receptors in peripheral tissues. The compound demonstrates long-acting antihistaminic activity with minimal anticholinergic effects in cellular assays. Studies investigate its role in mast cell degranulation inhibition and inflammatory mediator release modulation. Comparative research evaluates desloratadine against other compounds available in our desloratadine research collection. Scientists also examine its pharmacokinetic properties, including hepatic metabolism via CYP3A4 and CYP2D6 pathways. Research applications extend to investigating histamine’s role in various physiological processes and allergic response mechanisms. Laboratory studies analyse the compound’s selectivity profile compared to first and second-generation antihistamines. Advanced research explores desloratadine’s potential anti-inflammatory properties beyond traditional H1 receptor antagonism, including effects on cytokine release and immune cell activation pathways. Researchers studying similar receptor systems often cross-reference findings with SARM receptor research and peptide signaling studies.
Technical Specifications
| Parameter | Specification |
|---|---|
| Active Compound | Desloratadine |
| Manufacturer | Intas Pharmaceuticals |
| Strength | 5 mg per tablet |
| CAS Number | 100643-71-8 |
| Molecular Formula | C₁₉H₁₉ClN₂ |
| Molecular Weight | 310.82 g/mol |
| Storage Conditions | Room temperature, dry environment |
| Research Grade | Pharmaceutical standard |
Compliance Statement
Dezlorid 5 mg is supplied exclusively for in-vitro laboratory research purposes. This product is not intended for human consumption, therapeutic use, or any clinical applications. Researchers must ensure appropriate laboratory safety protocols and regulatory compliance when conducting studies with this material. All research activities should be performed by qualified personnel in controlled laboratory environments with proper documentation and safety measures.
